SCIENCE CHINA Chemistry 有机合成合辑

Virtual Issue: Organic Synthesis 

2018

Perspective

Synthetic porphyrin chemistry in China

Chengjie Li, Junlong Zhang, Jianxin Song, Yongshu Xie, Jianzhuang Jiang

Sci. China Chem., 2018, 61(5): 511-514 

Reviews

Recent developments in peptide ligation independent of amino acid side-chain functional group

Jinhua Yang, Junfeng Zhao

Sci. China Chem., 2018, 61(1): 97-112

Total chemical and semisynthetic approaches for the preparation of ubiquitinated proteins and their applications

Xiaobao Bi, Kumar Kalyan Pasunooti, Chuan-Fa Liu

Sci. China Chem., 2018, 61(3): 251-265

Feature Article

Recent advances in Ni−Al bimetallic catalysis for unreactive bond transformation

Yin-Xia Wang & Mengchun Ye

Sci. China Chem., 2018, 61(8): 1004–1013

Communications

Ruthenium(II)-catalyzed synthesis of phthalides via the cascade addition and cyclization of aromatic acids with aldehydes

Juan Fan, Peng-Min Wang, Jia-Ni Wang, Xue Zhao, Zhong-Wen Liu, Jun-Fa Wei, Xian-Ying Shi

Sci. China Chem., 2018, 61(2): 153-158

Highly enantioselective cyclopropanation of tri-substituted olefins

Jun Li, Long Zheng, Hao Chen, Lijia Wang, Xiu-Li Sun, Jun Zhu, Yong Tang

Sci. China Chem., 2018, 61(5): 526-530

Phosphineoxide-Sc(OTf)₃ catalyzed enantioselective bromoaminocyclization of tri-substituted allyl N-tosylcarbamates

Xiangyu Tan, Hongjie Pan, Hua Tian, Yian Shi

Sci. China Chem., 2018, 61(6): 656-659

Cu(II)-catalyzed aerobic oxidative amidation of azoarenes with amides

Gang Li, Xiaoting Chen, Xulu Lv, Chunqi Jia, Panpan Gao, Ya Wang, Suling Yang

Sci. China Chem., 2018, 61(6): 660-663

Probing guest compounds enabling the facile isolation of cucurbit[10]uril

Xiran Yang, Zhiyong Zhao, Xiongzhi Zhang, Simin Liu

Sci. China Chem., 2018, 61(7): 787-791

Oxidation-induced ortho-selective C–H bond functionalization of 2-naphthylamine derivative

Dongchao Zhang, Zhiliang Huang & Aiwen Lei

Sci. China Chem., 2018, 61(10): 1274–1277 

Articles

C(sp3)–H bond functionalization of non-cyclic ethers by decarboxylative oxidative coupling with α,β-unsaturated carboxylic acids

Tong Zhang, Xing-Wang Lan, Yu-Qiang Zhou, Nai-Xing Wang, Yue-Hua Wu, Yalan Xing, Jia-Long Wen

Sci. China Chem., 2018, 61(2): 180-183 

Oxygen as an oxidant in rhodium(III) catalyzed oxidative C–H/C–H cross-coupling between indoles and oxazoles

Yan Wang, Jingbo Lan

Sci. China Chem., 2018, 61(2): 200-205

Visible light-promoted, iodine-catalyzed selenoalkoxylation of olefins with diselenides and alcohols in the presence of hydrogen peroxide/air oxidant: an efficient access to α-alkoxyl selenides 

Mingxuan Liu, Yiming Li, Lei Yu, Qing Xu, Xuefeng Jiang

Sci. China Chem., 2018, 61(3): 294-299 

Semi-synthesis of disulfide-linked branched tri-ubiquitin mimics

Yanyan Si, Lujun Liang, Shan Tang, Yunkun Qi, Yong Huang, Lei Liu

Sci. China Chem., 2018, 61(4): 412-417 

Discovery of natural berberine-derived nitroimidazoles as potentially multi-targeting agents against drug-resistant Escherichia coli

Guo-Biao Zhang, Kameswari Swetha Maddili, Vijai Kumar Reddy Tangadanchu, Lavanya Gopala, Wei-Wei Gao, Gui-Xin Cai, Cheng-He Zhou

Sci. China Chem., 2018, 61(5): 557-568 

Metal-free synthesis of quinolines by direct condensation of amides with alkynes: revelation of N-aryl nitrilium intermediates by 2D NMR techniques 

Jian-Liang Ye, Ya-Nan Zhu, Hui Geng, Pei-Qiang Huang

Sci. China Chem., 2018, 61(6): 687-694

Palladium-catalyzed oxidative cyclopropanation of enamides and norbornenes initiated by C–H activation

Ming Chen, Mi-Na Zhao, Yao-Du Zhang, Zhi-Hui Ren, Zheng-Hui Guan

Sci. China Chem., 2018, 61(6): 695-701

Racemic X-ray structure of L-type calcium channel antagonist Calciseptine prepared by total chemical synthesis

Chen-Chen Chen, Shuai Gao, Hua-Song Ai, Qian Qu, Chang-Lin Tian, Yi-Ming Li

Sci. China Chem., 2018, 61(6): 702-707

A convenient method to prepare random LA/CL copolymers from poly(L-lactide) and ε-caprolactone

Hao Ouyang, Kun Nie, Dan Yuan, Yong Zhang, Dongmei Cui, Yingming Yao

Sci. China Chem., 2018, 61(6): 708-714

A stable metal-covalent-supramolecular organic framework hybrid: enrichment of catalysts for visible light-induced hydrogen production

Xiong-Fei Li, Shang-Bo Yu, Bo Yang, Jia Tian, Hui Wang, Dan-Wei Zhang, Yi Liu, Zhan-Ting Li

Sci. China Chem., 2018, 61(7): 830-835

A new class of HIV-1 inhibitors and the target identification via proteomic profiling

Ying-Zi Ge, Bin Zhou, Ruo-Xuan Xiao, Xiao-Jing Yuan, Hu Zhou, Ye-Chun Xu, Mark A. Wainberg,Ying-Shan Han & Jian-Min Yue

Sci. China Chem., 2018, 61(11): 1430–1439

Metal-free visible-light-mediated aerobic oxidation of silanes to silanols

Jing Wang, Bin Li, Li-Chuan Liu, Chenran Jiang, Tao He& Wei He

Sci. China Chem., 2018, 61(12): 1594–1599

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2017

Minireviews

N-cap helix nucleation: methods and their applications

Dongyuan Wang, Xuan Qin, Hui Zhao & Zigang Li

Sci. China Chem., 2017, 60(6): 689–700

Ni-mediated C–N activation of amides and derived catalytic transformations

Yuan Gao, Chong-Lei Ji & Xin Hong

Sci. China Chem., 2017, 60(11): 1413–1424

Reviews

Recent advances in the preparation of Fmoc-SPPS-based peptide thioester and its surrogates for NCL-type reactions

Hongxing Li & Suwei Dong

Sci. China Chem., 2017, 60(2): 201–213

Recent advances in radical-mediated fluorination through C–H and C–C bond cleavage

Hong Yan & Chen Zhu

Sci. China Chem., 2017, 60(2): 214–222

Recent advances in direct dehydrogenative biphenyl couplings

Fei Lv & Zhu-Jun Yao

Sci. China Chem., 2017, 60(6):701–720

Recent progress on the synthesis of 2-deoxy glycosides

Jing Zeng, Yang Xu, Hao Wang, Lingkui Meng & Qian Wan

Sci. China Chem., 2017, 60(9): 1162–1179

Communications

Metal-free tetra-n-butylammonium bromide-mediated aerobic oxidative synthesis of β-ketosulfones from styrenes using unnatural amino acids

Xin Wan, Kai Sun & Guisheng Zhang

Sci. China Chem., 2017, 60(3): 353–357

Direct access to β-seleno sulfones at room temperature through selenosulfonylation of alkenes

Kai Sun, Yunhe Lv, Zuodong Shi, Fangfang Fu, Chong Zhang & Zhiguo Zhang

Sci. China Chem., 2017, 60(6): 730–733

Articles

PhI(OAc)2-promoted umpolung acetoxylation of enamides for the synthesis of α-acetoxy ketones

Ming Chen, Wei Zhang, Zhi-Hui Ren, Wen-Yun Gao, Yao-Yu Wang & Zheng-Hui Guan

Sci. China Chem., 2017, 60(6): 761–768

Design, synthesis and biological evaluation of amino organophosphorus imidazoles as a new type of potential antimicrobial agents

Wei-Wei Gao, Syed Rasheed, VijaiKumar Reddy Tangadanchu, Yi Sun, Xin-Mei Peng, Yu Cheng, Feng-Xiu Zhang, Jian-Mei Lin & Cheng-He Zhou

Sci. China Chem., 2017, 60(6): 769–785